Discovery and development of antiandrogens Testosterone/dutasteride Drupanol MK-3984 Polytestosterone phloretin phosphate Linuron BOMT Inocoterone LG121071 DIMP (antiandrogen) Andarine Testosterone acetate butyrate 5N-Bicalutamide Methylhydroxynandrolone Cyanonilutamide JNJ-28330835 Δ4-Abiraterone RD-162 Methylclostebol RU-22930 Vinyltestosterone Testosterone acetate propionate GSK2881078 RU-58642 AA560 18-Methyltestosterone LGD-2941 OPK-88004 N-Desmethylapalutamide Pentomone Ralaniten Pyrilutamide Acetothiolutamide Benorterone ACP-105 GLPG-0492 Testosterone formate Chlorodehydromethylandrostenediol Ketodarolut…
tamide 1-Androstenedione Dienedione PF-06260414 Vosilasarm Testosterone dipropionate RU-59063 Topterone Metogest 4-Hydroxytestosterone Mesterolone cipionate Dihydrofluoxymesterone Testosterone isovalerate N-Desmethylenzalutamide Ethyldienolone Methyldienolone RU-58841 3-Keto-5α-abiraterone 19-Norandrosterone S-23 (drug) Procymidone LGD-3303 GSK-4336A Inocoterone acetate LG-120907 Plomestane 1-Androstenediol LGD-2226 Rezvilutamide Boldione BMS-564,929 RU-56187 Cioteronel Ligandr
ol Atraric acid S-40503 Delanterone AC-262,536 4-Dehydroepiandrosterone Chloromethylandrostenediol Rosterolone Proxalutamide Allyltestosterone RU-57073 Masofaniten Dimethylcurcumin Dihydrotestosterone butyrate Methasterone Dihydrotestosterone acetate Dihydrotestosterone undecanoate YK-11 Methyldiazinol Sturamustine Oxofluoxymesterone 7α-Methyl-19-norandrostenedione Methylstenbolone 5α-Dihydronandrolone Testosterone phenylbutyrate Nordinone Stenbolone Desoxymethyltestosterone Methandriol diacetate Norboletone Enestebol 1-Testosterone TFM-4AS-1 5α-Androst-2-ene-17-one EC586 Acetoxolutamide Bolenol Clascoterone Cl-4AS-1 Ethyltes
Testosterone/dutasteride
Drupanol
MK-3984
Polytestosterone phloretin phosphate
Linuron
BOMT
Inocoterone
LG121071
DIMP (antiandrogen)
Andarine
Testosterone acetate butyrate
5N-Bicalutamide
Methylhydroxynandrolone
Cyanonilutamide
JNJ-28330835
Δ4-Abiraterone
RD-162
Methylclostebol
RU-22930
Vinyltestosterone
Testosterone acetate propionate
GSK2881078
RU-58642
AA560
18-Methyltestosterone
LGD-2941
OPK-88004
N-Desmethylapalutamide
Pentomone
Ralaniten
Pyrilutamide
Acetothiolutamide
Benorterone
ACP-105
GLPG-0492
Testosterone formate
Chlorodehydromethylandrostenediol
Ketodarolutamide
1-Androstenedione